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Bioinformatics and drug discovery /edited by Richard S. Larson --Humana Press, 2006. --(58.17/M592/v.316)

Contents

Contents:

1. New Strategies in Drug Discovery  1

2. Basic Microarray Analysis: Strategies for Successful Experiments  13

3. From Microarray to Biological Networks: Analysis of Gene Expression

    Profiels  35

4. Microarray Analysis in Drug Discovery and Clinical Applications  49

5.Ontology-Driven Approaches to Analyzing Data in Functional Genomics  67

6. Gene Evolution and Drug Discovery  87

7. Standardization of Microarray and Pharmacogenomics Data  111

8. Clinical Applications of Bioinformatics, Genomics, and

     Pharmacogenomics  159

9. Protein Interactions Probed With Mass Spectrometry  179

10. Discovering New Drug-Targeting Sites on Flexible Multidomain Protein

      Kinases: Combing Segmental Isotopic and Site-Directed Spin Labeling for

      Nuclear Magnetic Resonance Dectection of Interfacial Clefts  199

11. Nuclear Magnetic Resonance-Based Screening Methods for Drug 

      Discovery  227

12. Receptor-Binding Sites: Bioinformatic Approaches  291

13. In Silico Protein Design: Fitting Sequence Onto Structure  359

14. Chemical Database Preparation for Compound Acquisition or

       Virtual  Screening  375

15. Bioinformatics Platform Development: From Gene to lead Compound  389