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Contemporary drug synthesis / by Jie Jack Li ... [et al.]. -- Wilety-Interscience, 2004. -- 63.326/C761

Contents

Contents:

1. Antithrombotics: Ticlopidine (Tielid) and Clopidogrel (Plavix)  1

2. Anti-inflammatory Cyclooxygenase-2 Selective Inhibitors : Celecoxib (Celebrex) and Rofecoxib (Vioxx)  11

3. H(+)/K(+)-ATPase Inhibitors: Esomeprazole (Nexium)  21

4. Protein-tyrosine Kinase Inhibitors: Imatinib (Gleevec) and Gefitinib (Iressa)  29

5. Non-sedating Antihistamines  39

6. Cosmeceuticals: Isotretinoin (Accutane), Tazarotene (Tazorac) Minoxidil (Rogaline), and Finasteride (Propecia)  55

7. antivacterials: Ciprofloxacin (Cipro) and Linezolid (Zyvox)  75

8. Atypical antipsychotics  89

9. Atorvastatin Calcium (Lipitro)  113

10. Antidepressants  125

11. anti-obesity: Orlistat (Xenical)  149

12. Triptans for Migraine  161

13. PDE 5 Inhibitors for Erectile Dysfunction: Sidebafil (Viagra), Vardenafil (Levitra) , and Tadalafil (Cialis)  189

14. Antiasthmatics  201